Cart
sales@molnova.com
CBiPES hydrochloride
CAS No. 856702-40-4
CBiPES hydrochloride( —— )
Catalog No. M33836 CAS No. 856702-40-4
CBiPES hydrochloride (CBiPES HCl) is a potent orthosteric modulator of the mGlu2 receptor with an EC50 value of 92.8 nM.CBiPES hydrochloride blocks the action of WT and mGlu(3) receptors.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 263 | Get Quote |
|
| 5MG | 416 | Get Quote |
|
| 10MG | 603 | Get Quote |
|
| 25MG | 906 | Get Quote |
|
| 50MG | 1214 | Get Quote |
|
| 100MG | 1611 | Get Quote |
|
| 500MG | 3231 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameCBiPES hydrochloride
-
NoteResearch use only, not for human use.
-
Brief DescriptionCBiPES hydrochloride (CBiPES HCl) is a potent orthosteric modulator of the mGlu2 receptor with an EC50 value of 92.8 nM.CBiPES hydrochloride blocks the action of WT and mGlu(3) receptors.
-
DescriptionCBiPES hydrochloride is a mGlu2 receptor positive allosteric modulator (EC50: 92.8 nM). CBiPES hydrochloride attenuates stress-induced hyperthermia and PCP-induced hyperlocomotor activity. CBiPES hydrochloride can be used for research of neurological disease.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayNeuroscience
-
TargetGluR
-
RecptorGluR
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number856702-40-4
-
Formula Weight413.92
-
Molecular FormulaC21H20ClN3O2S
-
Purity>98% (HPLC)
-
Solubility——
-
SMILESCl.N#CC1=CC=C(C=C1)C=2C=CC=C(C2)N(CC=3C=NC=CC3)S(=O)(=O)CC
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Johnson MP, et al. Metabotropic glutamate 2 receptor potentiators: receptor modulation, frequency-dependent synaptic activity, and efficacy in preclinical anxiety and psychosis model(s). Psychopharmacology (Berl). 2005 Apr;179(1):271-83.?
molnova catalog
related products
-
S 18986
S 18986 is a selective, orally active, brain-penetrant positive allosteric modulator of AMPA-type receptors that enhances cognition in rodents by inducing the release of noradrenaline and acetylcholine in the rat hippocampus, subsequently improving object-recognition memory.
-
KML29
KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor.
-
HBT1
HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons. HBT1 binds to ligand-binding domain of AMPA-R in glutamate dependent manner.HBT1 bound to the ligand-binding domain (LBD) of AMPA-R in a glutamate-dependent manner.?
